Adrenergic agonists
Direct acting
alpha-1 (A,B,C,D) adrenergic receptors (selective agonists)
- Metoxamine
- Phenylephrine
- Naphazoline
- Oximethazoline
alpha-2 (A,B,C) adrenergic receptors (selective agonists)
- Alpha methyldopa
- Brimonidine
- Clonidine
- Guanfacine
beta (1,2,3) adrenergic receptors (selective agonists)
- Salbutamol (2)
- Fomoterol (2)
- Doutamine (1)
alpha-1 (A,B,C,D); alpha-2 (A,B,C); beta(1,2,3) (non-selective agonists)
- Epinephrine (Adrenaline)
- Norepinephrine (Noradrenaline)
Mixed acting
- Ephedrine
Indirect acting
- Selegiline
- Entecapone
alpha (A,B,C,D); alpha-2 (A,B,C); beta (1,2,3) (non-selective agonists)
- Amphetamine
Adrenergic antagonists (Antiadrenergics)
alpha-1 (A,B,C,D); alpha-2 (A,B,C); beta (1,2,3) (selective agonists)
- Pranzosin
- Doxazosin
- Terazosin
alpha-2 (A,B,C) adrenergic receptors (selective antagonist)
- Yohimbine
beta (1) adrenergic receptors (non-selective antagonists) [First generation]
- Pindolol
- propanolol
- Nadolol
- Timolol
beta (1) adrenergic receptors (selective antagonists) [Second Generation]
- Atenolol
- Esmolol
alpha-1 (A,B,C,D); alpha-2 (A,B,C); beta (1,2,3) (non-selective antagonists) [Third generation]
- Carvedilol
- Labetolol